Tracer | LogD7.4 (n = 3) | Intact fraction (%) in plasma at 15 min post-injection |
---|---|---|
[68Ga]Ga-TacBOMB2 | − 3.21 ± 0.04 | 12.7 ± 2.93 |
[68Ga]Ga-LW01107 | − 3.10 ± 0.05 | 66.2 ± 12.4 |
[68Ga]Ga-LW01108 | − 3.10 ± 0.02 | 35.3 ± 0.93 |
[68Ga]Ga-LW01110 | − 2.83 ± 0.08 | 89.0 ± 2.17 |
[68Ga]Ga-LW01142 | − 1.81 ± 0.02 | 91.2 ± 5.30 |
[68Ga]Ga-LW02021 | − 2.46 ± 0.09 | – |
[68Ga]Ga-LW02040 | − 2.48 ± 0.12 | 92.9 ± 2.30 |
[68Ga]Ga-RM2 | − 2.76 ± 0.03 | 71.9 ± 10.4 |
[68Ga]Ga-AMBA | − 3.66 ± 0.03 | 39.4 ± 10.8 |