derivative | Ki ± SD / nM | Internalization ± SD / %IA/106 cells | ||
---|---|---|---|---|
[nat/68Ga]Ga-PSMA-11 | 12.0 ± 2.8 | (Eder et al. 2012a) | 9.5 ± 2.6 | (Benešová et al. 2015) |
[nat/68Ga]Ga-PSMA-617 | 6.4 ± 1.0 | (Benešová et al. 2015) | 17.7 ± 4.4 | (Benešová et al. 2015) |
[nat/68Ga]Ga-AAZTA5-PSMA | 8.7 ± 0.9 | 13.0 ± 0.2 | ||
[nat/44Sc]Sc-PSMA-617 | 4.7 ± 0.8 | (Eppard et al. 2017) | 15.8 ± 2.1 | (Eppard et al. 2017) |
[nat/44Sc]Sc-AAZTA5-PSMA | 30.6 ± 11.5 | 20.0 ± 0.9 | ||
[nat/177Lu]Lu-PSMA-617 | 6.9 ± 1.3 | (Benešová et al. 2015) | 17.5 ± 3.1 | (Benešová et al. 2015) |
[nat/177Lu]Lu-AAZTA5-PSMA | 26.6 ± 11.1 | 18.0 ± 2.0 |