Compound | IC50 [nM] |
---|---|
FC131 | 9.9 ± 2.4a |
[natGa]pentixafor (DOTA) | 24.8 ± 2.5a |
[natCu]DOTAGA-pentixafor | 1165 ± 220a |
[natCu]NOTA-pentixafor | 46.1 ± 26a |
[natCu]NODAGA-pentixafor | 343 ± 10a |
[natCu]DTPA-pentixafor | 175 ± 66a |
NOTA-pentixather | 27.5 ± 2.1 |
[natCu]NOTA-pentixather | 14.9 ± 2.1 |
NODAGA-pentixather | 64.9 ± 6.5 |
[natCu]NODAGA-pentixather | 47.5 ± 1.8 |